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ЗАМІЩЕНІ ПІРИДОПІРАЗИНИ ЯК ІНГІБІТОРИ Syk

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(11)
111744
(22)
07.06.2012
(24)
10.06.2016
(21)
a201315617
(31)
PCT/CN2011/075431
(32)
08.06.2011
(33)
CN
(41)
12.05.2014, бюл. № 9
(46)
10.06.2016, бюл. № 11
(56)
WO 2004005472 (A2), 15.01.2004
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CARROLL TEMPLE, JR. ET AL.: "1,2-Dihydropyrido[3,4-b] pyrazines: Structure-Activity Relationships.", J. MED. CHEM., vol. 26, no. 1, 1983, pages 91-95
JEFFREY W. WILLIAMS ET AL.: "The inhibition of dihydrofolate reductase by folate analogues: structural requirements for slow- and tight-binding inhibition.", BIOCHEMICAL PHARMACOLOGY, vol. 29, no. 4, 1980, pages 589-595
BRITTA NISIUS ET AL.: "Development of a Fingerprint Reduction Approach for Bayesian Similarity Searching Based on Kullback-Leibler Divergence Analysis.", J. CHEM. INF. MODEL., vol. 49, no. 6, 2009, pages 1347-1358
ROBERT D. ELLIOTT ET AL.: "Potential Folic Acid Antagonists. VI. The Syntheses of 1- and 3-Deazamethotrexate.", J. ORG. CHEM., vol. 36, no. 19, 1971, pages 2818-2823
C. CHOO HOFFMANN ET AL.: "Comparative effects of selected antifolates on transforming human lymphocytes and on established human lymphoblastic cell lines.", BIOCHEMICAL PHARMACOLOGY, vol. 25, no. 17, 1976, pages 1947-1954
DELIANG CHEN ET AL.: "Computational Selection of Inhibitors of A-beta Aggregation and Neuronal Toxicity.", BIOORG MED CHEM., vol. 17, no. 14, 15 July 2009 (2009-07-15), pages 5189-5197
ROBERT D. ELLIOTT ET AL.: "The Isomeric Pyridopyrazines from the Reaction of Some Tetraaminopyridines with Pyruvaldehyde and Benzil.", THE JOURNAL OF ORGANIC CHEMISTRY, vol. 33, no. 6, June 1968, pages 2393-2397
(85)
08.01.2014
(86)
PCT/CN2012/076576, 07.06.2012
(71)
ХАТЧІСОН МЕДІФАРМА ЛІМІТЕД CN
 
HUTCHISON MEDIPHARMA LIMITED CN
(72)
Су Вей-Го CN; Ден Вей CN; Цзі Цзяньго CN
 
Su, Wei-Guo CN; Deng, Wei CN; Ji, Jianguo CN
(73)
ХАТЧІСОН МЕДІФАРМА ЛІМІТЕД CN
 
HUTCHISON MEDIPHARMA LIMITED CN
(74)
Михайлюк Валентин Іванович
(98)
Михайлюк Валентин Iванович
вул. Бобруйська, 46, м. Харкiв, 61054, Україна
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